[Version 7General-EMEA/182460/2007 Wojtylová Jana722005-07-27T07:58:00Z2009-01-22T10:23:00Z2020-11-12T09:49:00Z1198711724Translation Centre19302497271368414General-EMEA/182460/2007V01a CS SPC-II-lab-pl v 7.1Holemarova Zuzana23/04/2007 10:24:26Holemarova ZuzanaHolemarova Zuzana23/04/2007 10:24:26emea_document0.2, CURRENT, published April 07EMEA/182460/2007182460nulldateGeneralEMEAnulldate2007nulldatePŘÍLOHA ISOUHRN ÚDAJŮ O PŘÍPRAVKU1.NÁZEV VETERINÁRNÍHO LÉČIVÉHO PŘÍPRAVKUEffipro duo 100 mg/120 mg roztok pro nakapání na kůži – spot-on pro velmi velké kočky2.KVALITATIVNÍ A KVANTITATIVNÍ SLOŽENÍPipeta (1 ml) obsahuje:Léčivé látky:Fipronilum 100 mgPyriproxyfenum 120 mgPomocné látky:Butylhydroxyanisol (E 320) 0,2 mgButylhydroxytoluen (E 321) 0,1 mgÚplný seznam pomocných látek viz bod 6.1.3.LÉKOVÁ FORMARoztok pro nakapání na kůži – spot-on.Čirý, bezbarvý až nažloutlý roztok.4.KLINICKÉ ÚDAJE4.1Cílové druhy zvířatKočky (>6-12 kg).4.2Indikace s upřesněním pro cílový druh zvířatLéčba napadení koček blechami samostatně nebo ve spojení s klíšťaty.Proti blechám:Léčba a prevence napadení blechami (Ctenocephalides felis). Jedno ošetření zabrání další infestaci po dobu 5 týdnů.Prevence množení blech prostřednictvím přerušení vývoje vajíček v dospělé blechy po dobu 12 týdnů po aplikaci.Přípravek může být použit jako součást léčebné strategie při zvládání alergické dermatitidy po bleším kousnutí (FAD), která byla předtím diagnostikována veterinárním lékařem.Proti klíšťatům:Léčba napadení klíšťaty (Ixodes ricinus a Rhipicephalus turanicus). Jedno ošetření poskytuje trvalý akaricidní účinek po dobu jednoho týdne. Pokud jsou klíšťata v době aplikace přítomna, je možné, že nebudou všechna v průběhu 48 hodin usmrcena.4.3KontraindikaceNepoužívat u králíků z důvodu možného výskytu nežádoucích účinků nebo až úhynu.Nepoužívat v případě známé přecitlivělosti na léčivé látky nebo na některou z pomocných látek.4.4Zvláštní upozornění pro každý cílový druhNamáčení srsti vodou dvě hodiny před aplikací přípravku a dvakrát během uvedené doby účinnosti proti blechám (ve dvoutýdenních intervalech proti dospělým blechám nebo čtyřtýdenních intervalech proti vývojovým stádiím blech) bylo zkoumáno ve dvou laboratorních studiích. Namáčení srsti vodou tak, jak je popsáno výše, nemělo nepříznivý vliv na účinnost přípravku.Vliv šamponování na účinnost přípravku nebyl zkoumán. Pokud však je u kočky šamponování potřebné, doporučuje se jeho provedení před aplikací veterinárního léčivého přípravku.Na počátku léčebných opatření v případě infestace by měly být přepravky zvířat a místa, kde zvířata spí a odpočívají, jako jsou koberce a bytové zařízení, pravidelně ošetřovány vhodným insekticidem a vysávány. Aby se snížilo množství blech v prostředí, je třeba ošetřit vhodným přípravkem proti blechám veškerá zvířata žijící ve stejné domácnosti.Přípravek nebrání přichycení klíšťat ke zvířeti. Pokud bylo zvíře ošetřeno předtím, než přišlo do styku s klíšťaty, budou klíšťata usmrcena do 48 hodin po přichycení. To obvykle nastane před jejich zvětšením nasátím, což minimalizuje, ale nevyloučí riziko přenosu chorob.Uhynulá klíšťata většinou sama odpadávají ze zvířete. Jakákoliv zbylá klíšťata by měla být opatrně odstraněna tak, aby jejich ústní ústrojí nezůstalo v kůži zvířete.4.5Zvláštní opatření pro použitíZvláštní opatření pro použití u zvířat:Jen pro zevní použití. Nepodávejte perorálně. Před ošetřením by měla být zvířata přesně zvážena. Nebyla stanovena bezpečnost přípravku u koťat mladších 10 týdnů nebo u koček o hmotnosti nižší než 1 kg. Zabraňte kontaktu s očima zvířete. V případě náhodného zasažení očí je vypláchněte vodou. Je třeba dbát na to, aby byl přípravek aplikován přesně podle popisu v bodě 4.9. Neaplikovat přípravek na rány nebo poraněnou kůži. Je důležité zabezpečit, aby byl veterinární léčivý přípravek aplikován přímo na suchou kůži v místě, kde si jej zvíře nemůže olízat, a také, aby si jej zvířata po ošetření nemohla olízat navzájem.Použití přípravku nebylo zkoumáno u oslabených nebo nemocných koček. U nemocných nebo oslabených zvířat použít pouze po zvážení poměru terapeutického prospěchu a rizika příslušným veterinárním lékařem.Vzhledem k absenci dalších studií týkajících se bezpečnosti přípravku, neopakovat ošetření v intervalech kratších než 4 týdny.Zvláštní opatření určené osobám, které podávají veterinární léčivý přípravek zvířatům:Přípravek může působit neurotoxicky. Při požití může být přípravek škodlivý.Zabraňte požití, včetně kontaktu rukou s ústy.Během aplikace přípravku nekuřte, nepijte ani nejezte.V případě náhodného požití vyhledejte ihned lékařskou pomoc a ukažte příbalovou informaci nebo etiketu praktickému lékaři.Tento přípravek může způsobit podráždění očí a sliznic.Zabraňte kontaktu s kůží, očima a ústy, včetně kontaktu rukou s očima.V případě náhodného kontaktu s kůží nebo očima ihned důkladně opláchněte postižené místo vodou. Pokud podráždění kůže nebo očí přetrvává, vyhledejte lékařskou pomoc a ukažte příbalovou informaci nebo etiketu lékaři.Po použití si umyjte ruce.Nemanipulujte s ošetřenými zvířaty a zamezte dětem hrát si s nimi, dokud místo aplikace nezaschne. Doporučuje se proto neošetřovat zvířata během dne, ale v podvečer, a nedovolit čerstvě ošetřeným zvířatům spát s jejich majiteli, zejména s dětmi. Uchovávejte pipety v původním obalu až do doby použití a poté je ihned zlikvidujte.Další opatřeníPřípravek může mít nepříznivý vliv na natřené, lakované nebo jiné plochy v domácnosti nebo vybavení bytu. Před kontaktem s takovými materiály nechte místo aplikace zaschnout.4.6Nežádoucí účinky (frekvence a závažnost)V místě aplikace se mohou objevit přechodné kosmetické změny, jako například mokrý vzhled srsti nebo mírná tvorba lupů. Nashromážděné údaje o těchto léčivých látkách ve formě spot-on přípravků ukazují, že se po použití mohou v místě aplikace objevit přechodné kožní reakce (tvorba šupin na kůži, lokální alopecie, pruritus, erytém, změny barvy srsti) a celkový pruritus nebo alopecie. Mohou se vyskytnout hypersalivace, reversibilní neurologické symptomy (hyperesthesie, deprese, nervové příznaky), dýchací příznaky nebo zvracení. Tyto příznaky se vyskytují ve velmi vzácných případech.Četnost nežádoucích účinků je charakterizována podle následujících pravidel:- velmi časté (nežádoucí účinek(nky) se projevil(y) u více než 1 z 10 ošetřených zvířat)- časté (u více než 1, ale méně než 10 ze 100 ošetřených zvířat)- neobvyklé (u více než 1, ale méně než 10 z 1000 ošetřených zvířat)- vzácné (u více než 1, ale méně než 10 z 10000 ošetřených zvířat)- velmi vzácné (u méně než 1 z 10000 ošetřených zvířat, včetně ojedinělých hlášení).4.7Použití v průběhu březosti, laktace a snáškyLaboratorní studie s fipronilem a pyriproxyfenem neprokázaly teratogenní nebo embryotoxický účinek. Bezpečnost přípravku u březích a laktujících koček nebyla stanovena. Ošetření v březosti a laktaci by mělo být provedeno pouze po zvážení poměru terapeutického prospěchu a rizika příslušným veterinárním lékařem.4.8Interakce s dalšími léčivými přípravky a další formy interakceNejsou známy.4.9Podávané množství a způsob podáníPoužití k nakapání na kůži – spot-on. Dávkování: Pro kočku o hmotnosti vyšší než 6 kg použijte jednu pipetu o objemu 1 ml, což odpovídá minimální doporučené dávce 8,3 mg fipronilu / kg živé hmotnosti a 10 mg pyriproxyfenu / kg ž. hm. Doporučené dávky 1 ml lze dosáhnout také použitím dvou pipet o objemu 0,5 ml. Hmotnost kočky Objem pipetyFipronil (mg)Pyriproxyfen (mg)6 – 12 kg 1 ml100120Způsob podání: Vyjměte pipetu z blistru. Držte pipetu svisle. Poklepejte na zúženou část pipety, abyste se ujistili, že obsah je uvnitř hlavní části pipety. Odlomte hrot pipety ve vyznačené linii. Rozhrňte srst zvířete na zadní části krku před lopatkami tak, aby byla viditelná kůže. 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Pro optimální zvládnutí napadení blechami a klíšťaty a množení blech by měl být režim ošetření založen na místní epidemiologické situaci. Vzhledem k absenci dalších studií týkajících se bezpečnosti přípravku, neopakovat ošetření v intervalech kratších než 4 týdny (viz bod 4.10).4.10Předávkování (symptomy, první pomoc, antidota), pokud je to nutnéVe studiích bezpečnosti pro cílové druhy zvířat vykonaných na 10 - týdenních koťatech, která byla léčena dávkou 5-ti násobně převyšující doporučenou dávku 3x v intervalech 4 týdnů a maximální doporučenou dávkou 6x v intervalech 4 týdnů, nebyly pozorovány žádné závažné nežádoucí účinky.Nebezpečí vzniku nežádoucích účinků (viz bod 4.6) se může zvýšit v případě předávkování, tudíž by zvířata měla být vždy ošetřena správnou velikostí pipety v závislosti na jejich živé hmotnosti.4.11Ochranná(é) lhůta(y)Není určeno pro potravinová zvířata. 5.FARMAKOLOGICKÉ VLASTNOSTIFarmakoterapeutická skupina: ektoparazitika pro lokální aplikaci, fipronil, kombinace.ATCvet kód: QP53AX65.5.1Farmakodynamické vlastnostiFipronil je insekticid a akaricid náležící do skupiny fenylpyrazolů. Fipronil a jeho metabolit fipronil sulfon působí na ligandem řízených chloridových kanálech, zejména těch řízených neurotransmiterem kyselinou gamaaminomáselnou (GABA), stejně jako desenzitizuje (D) a nedesenzitizuje (N) kanály řízené glutamátem (Glu, jedinečné ligandem řízené chloridové kanály bezobratlých), čímž blokuje pre- a postsynaptický přenos chloridových iontů přes buněčné membrány. Důsledkem toho je nekoordinovaná činnost centrálního nervového systému a úhyn hmyzu a roztočůPyriproxyfen je regulátor růstu hmyzu (IGR) ze skupiny látek známých jako analogy juvenilních hormonů. Pyriproxyfen sterilizuje dospělé blechy a brání vývoji nedospělých stádií. Kontakt s molekulou brání vzniku dospělců tím, že blokuje vývoj vajíček (ovicidní účinek), larev a kukel (larvicidní účinek), které jsou následně odstraněny. Po kontaktu s molekulou a/nebo pozření dospělou blechou též dochází ke sterilizaci vajíček v průběhu zrání ještě před jejich nakladením. Molekula předchází kontaminaci prostředí léčených zvířat nezralými vývojovými stádii blech. Kombinace fipronilu a pyriproxyfenu zajišťuje insekticidní a akaricidní účinek proti blechám (Ctenocephalides felis) a klíšťatům (Rhipicephalus turanicus, Ixodes ricinus) a navíc zabraňuje vývoji dospělých blech z vajíček. Tato kombinace poskytuje komplexní ochranu proti napadení blechami, která může být použita proti napadení blechami samostatně nebo ve spojení s klíšťaty. 5.2Farmakokinetické údaje Po topické aplikaci přípravku se za normálních podmínek použití fipronil a pyriproxyfen dobře distribuují v srsti od prvního dne po aplikaci. Hlavní metabolit fipronilu je sulfonový derivát, který má také insekticidní a akaricidní vlastnosti.Koncentrace fipronilu a pyriproxyfenu na srsti postupem času klesají, ale jsou stále detekovatelné po dobu nejméně 84 dní po aplikaci (tj. nad dolní mez stanovitelnosti (LOQ) 100 ng/g pro fipronil a 50 ng/g pro pyriproxyfen). Koncentrace fipronil sulfonu zůstaly pod dolní mezí stanovitelnosti (LOQ 100 ng/ml) po použití přípravku.Maximální plazmatické koncentrace fipronilu a pyriproxifenu je brzy dosaženo za 1 den po podání. Koncentrace fipronilu je měřitelná u všech koček do 3 dnů po podání (LOQ 1 ng/ml). Koncentrace pyriproxifenu je měřitelná u všech koček do 42 dnů po podání (LOQ 0,2 ng/ml). Koncentrace fipronil sulfonu zůstávají pod dolní mezí stanovitelnosti (LOQ 1 ng/ml) po použití přípravku.6.FARMACEUTICKÉ ÚDAJE6.1Seznam pomocných látekButylhydroxyanisol (E 320)Butylhydroxytoluen (E 321)Diethylenglykol-monoethylether6.2Hlavní inkompatibilityNejsou známy.6.3Doba použitelnostiDoba použitelnosti veterinárního léčivého přípravku v neporušeném obalu: 3 roky. 6.4Zvláštní opatření pro uchováváníUchovávejte při teplotě do 30 °C. Uchovávejte v suchu. Uchovávejte blistr v krabičce, aby byl chráněn před světlem.6.5Druh a složení vnitřního obaluPrůhledné vícevrstvé plastové jednodávkové pipety s obsahem 1 ml vyrobené tepelným tvarováním spodní části (polyakrylonitrilmetakrylát nebo polyethylen-ethylen vinyl alkohol-polyethylen, polypropylen, kopolymer cyklického olefinu, polypropylen) a uzavřené tepelným svařením a víčkem (polyakrylonitrilmetakrylát nebo polyethylen-ethylen vinyl alkohol-polyethylen, hliník, polyethylentereftalát). Krabičky obsahují jednotlivé pipety umístěné v blistrových přebalech vyrobených z polypropylenu, kopolymeru cyklického olefinu, polypropylenu a uzavřených víčkem vyrobeným z polyethylentereftalátu, hliníku a polypropylenu.Krabičky po 1, 4, 24 nebo 60 pipetách (velké krabičky obsahují obálky určené pro vložení menšího počtu pipet). Na trhu nemusí být všechny velikosti balení.6.6Zvláštní opatření pro zneškodňování nepoužitého veterinárního léčivého přípravku nebo odpadu, který pochází z tohoto přípravkuVšechen nepoužitý veterinární léčivý přípravek nebo odpad, který pochází z tohoto přípravku, musí být likvidován podle místních právních předpisů. Přípravek nesmí kontaminovat vodní toky, protože může být nebezpečný pro ryby a další vodní organismy. Nekontaminujte rybníky, vodní toky nebo stoky přípravkem nebo prázdným obalem.7.DRŽITEL ROZHODNUTÍ O REGISTRACIVIRBAC1ère avenue – 2065m – LID06516 CarrosFRANCIE8.REGISTRAČNÍ ČÍSLO(A)96/065/16-C9.DATUM REGISTRACE/PRODLOUŽENÍ REGISTRACE8. 8. 2016/ 6. 10. 202010DATUM REVIZE TEXTUŘíjen 2020Velikost balení po 1 a 4 pipetách: Veterinární léčivý přípravek je vydáván bez předpisu. Vyhrazený veterinární léčivý přípravek.Velikost balení po 24 nebo 60 pipetách: Veterinární léčivý přípravek je vydáván pouze na předpis. PAGE \* MERGEFORMAT 7 PAGE \* MERGEFORMAT 1